SCHEMBL7230249

SCHEMBL7230249

COc1ccc2c(c1)-c1nc(Nc3cccc(NC=O)c3)ncc1CC2(C)C

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FYN P06241 2/20 0.56
KDR P35968 12/20 0.51
PLK1 P53350 10/20 0.51
INSR P06213 1/20 0.45
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
IKBKB O14920 1/20 0.44
IGF1R P08069 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7000614 0.85 KDR (0.64) FYNKDRPLK1INSRCCNA2
Hydrochloric Acid SCHEMBL6992934 0.84 FYN (0.54) FYNKDRPLK1INSRCCNA2
SCHEMBL6997719 0.84 FYN (0.58) FYNKDRPLK1INSRCCNA2
Hydrochloric Acid SCHEMBL7231258 0.83 FYN (0.54) FYNKDRPLK1INSRCCNA2
SCHEMBL6992927 0.82 FYN (0.58) FYNKDRPLK1INSRCCNA2
SCHEMBL7000795 0.82 FYN (0.56) FYNKDRPLK1CCNA2CDK2
Hydrochloric Acid SCHEMBL7238138 0.81 FYN (0.58) FYNKDRPLK1INSRCCNA2
SCHEMBL7235315 0.81 FYN (0.54) FYNKDRPLK1CCNA2CDK2
SCHEMBL7231388 0.81 FYN (0.61) FYNKDRPLK1INSRCCNA2
SCHEMBL7241122 0.81 FYN (0.65) FYNKDRPLK1INSRIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599908-B1 Potent and selective inhibitors of the protein tyrosine kinases p56lck and p59fyn CELLTECH R & D LIMITED (GB) 2003-07-29 US disclosed
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed