SCHEMBL7230278

SCHEMBL7230278

COc1cc(Nc2ncc3c(n2)-c2ccccc2CCC3)cc(OC)c1OC

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.67
IKBKB O14920 2/20 0.57
PTK2 Q05397 6/20 0.56
PLK1 P53350 2/20 0.50
PDGFRB P09619 2/20 0.50
JAK2 O60674 1/20 0.48
IGF1R P08069 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7241620 0.95 KDR (0.70) KDRIKBKBPTK2PLK1PDGFRB
SCHEMBL8035912 0.89 KDR (0.70) KDRPTK2PLK1PDGFRBJAK2
SCHEMBL7239285 0.83 KDR (0.63) KDRPTK2PLK1PDGFRBIGF1R
Hydrochloric Acid SCHEMBL7518134 0.83 KDR (0.62) KDRPTK2PLK1PDGFRBIGF1R
SCHEMBL7237418 0.82 FYN (0.65) KDRIKBKBPTK2PLK1PDGFRB
SCHEMBL7235444 0.82 IKBKB (0.67) KDRIKBKBPTK2PLK1PDGFRB
SCHEMBL7238442 0.81 KDR (0.60) KDRIKBKBPTK2PLK1PDGFRB
SCHEMBL7231942 0.81 KDR (0.58) KDRIKBKBPTK2PLK1PDGFRB
Hydrochloric Acid SCHEMBL7516453 0.81 IKBKB (0.66) KDRIKBKBPTK2PLK1PDGFRB
SCHEMBL7239325 0.81 KDR (0.58) KDRIKBKBPTK2PLK1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599908-B1 Potent and selective inhibitors of the protein tyrosine kinases p56lck and p59fyn CELLTECH R & D LIMITED (GB) 2003-07-29 US disclosed
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed