SCHEMBL8035912

SCHEMBL8035912

COc1cc(Nc2ncc3c(n2)-c2ccccc2C3)cc(OC)c1OC

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.70
PLK1 P53350 4/20 0.57
PTK2 Q05397 9/20 0.53
INSR P06213 2/20 0.52
AURKB Q96GD4 1/20 0.52
IGF1R P08069 2/20 0.50
JAK2 O60674 1/20 0.50
PDGFRB P09619 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7241620 0.91 KDR (0.70) KDRPLK1PTK2IGF1RJAK2
SCHEMBL7230278 0.89 KDR (0.67) KDRPLK1PTK2IGF1RJAK2
SCHEMBL7234789 0.81 KDR (0.64) KDRPLK1PTK2INSRAURKB
SCHEMBL7232394 0.81 KDR (0.64) KDRPLK1PTK2IGF1RJAK2
SCHEMBL7239285 0.81 KDR (0.63) KDRPLK1PTK2IGF1RPDGFRB
SCHEMBL7237382 0.81 KDR (0.63) KDRPLK1PTK2INSRAURKB
Hydrochloric Acid SCHEMBL7518134 0.80 KDR (0.62) KDRPLK1PTK2IGF1RPDGFRB
SCHEMBL7235444 0.80 IKBKB (0.67) KDRPLK1PTK2AURKBIGF1R
Hydrochloric Acid SCHEMBL7516453 0.79 IKBKB (0.66) KDRPLK1PTK2AURKBIGF1R
SCHEMBL7238442 0.79 KDR (0.60) KDRPLK1PTK2AURKBPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed