SCHEMBL7230776

SCHEMBL7230776

[O]Cc1cccc(F)c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.40
SLC6A4 P31645 3/20 0.39
SLC6A2 P23975 2/20 0.39
CYP2D6 P10635 1/20 0.39
KCNH2 Q12809 1/20 0.39
HCAR1 Q9BXC0 1/20 0.35
PTGS2 P35354 1/20 0.35
CMA1 P23946 5/20 0.34
TAAR1 Q96RJ0 1/20 0.34
LMNA P02545 1/20 0.33
TRPA1 O75762 1/20 0.33
IDO1 P14902 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12900215 0.83 GABRA1 (0.46) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL16701725 0.79 SLC6A4 (0.39) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL488379 0.79 SLC6A4 (0.39) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL19356887 0.79 SLC6A4 (0.39) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL488739 0.79 PDK2 (0.41) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL3166443 0.79 TAAR1 (0.43) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL27588706 0.78 GABRA1 (0.40) CYP2D6TAAR1LMNAGABRA1GABRB2
Hydrochloric Acid SCHEMBL2575776 0.78 TAAR1 (0.42) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL1541726 0.77 TRPA1 (0.40) P2RX7SLC6A4SLC6A2CYP2D6KCNH2
SCHEMBL27254254 0.76 SLC6A4 (0.40) P2RX7SLC6A4SLC6A2CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6544974-B2 Treating atherosclerosis and other coronary artery diseases. G.D. SEARLE & CO. 2003-04-08 US claimed