SCHEMBL7230934

SCHEMBL7230934

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1cnc(-c2cccc(O)c2)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.43
MAOA P21397 2/20 0.43
MAOB P27338 1/20 0.43
USP30 Q70CQ3 1/20 0.42
HSD17B1 P14061 5/20 0.42
HSD17B2 P37059 4/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MLLT1 Q03111 4/20 0.38
MLLT3 P42568 2/20 0.36
GSK3B P49841 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224277 0.89 USP30 (0.43) USP30HSD17B1HSD17B2NPC1POLB
SCHEMBL7223211 0.89 USP30 (0.41) USP30NPC1POLBRAB9ASMN1; SMN2
SCHEMBL7224212 0.89 USP30 (0.41) USP30NPC1POLBRAB9ASMN1; SMN2
SCHEMBL7226302 0.89 NPC1 (0.52) USP30CYP2C9NPC1POLBRAB9A
SCHEMBL7225292 0.89 P2RX7 (0.43) KDM1AMAOAMAOBUSP30NPC1
SCHEMBL7071274 0.89 USP30 (0.53) USP30CYP3A4CYP2C9NPC1RAB9A
Hydrochloric Acid SCHEMBL7075524 0.88 USP30 (0.52) USP30CYP3A4CYP2C9NPC1RAB9A
SCHEMBL7224996 0.88 USP30 (0.42) USP30HSD17B1HSD17B2NPC1RAB9A
SCHEMBL7232527 0.87 USP30 (0.42) USP30NPC1POLBRAB9ASMN1; SMN2
SCHEMBL7224838 0.87 USP30 (0.46) USP30CYP3A4NPC1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed