SCHEMBL7224838

SCHEMBL7224838

N#Cc1cccc(-c2ncc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.46
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
SLC6A2 P23975 2/20 0.39
SLC6A3 Q01959 2/20 0.39
AXL P30530 1/20 0.39
MERTK Q12866 1/20 0.39
PAX8 Q06710 1/20 0.39
CTSC P53634 1/20 0.38
HTR3A P46098 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
GRM5 P41594 2/20 0.36
CHEK1 O14757 5/20 0.36
PIM1 P11309 1/20 0.36
PLCG1 P19174 1/20 0.35
SLC6A4 P31645 1/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232113 0.89 USP30 (0.47) USP30CYP3A4CYP2D6CYP2C19SLC6A3
SCHEMBL7230934 0.87 KDM1A (0.43) USP30CYP3A4SLC6A3CHRNB2CHRNA4
SCHEMBL7224277 0.86 USP30 (0.43) USP30AXLMERTKCHRNB2CHRNA4
SCHEMBL7223211 0.86 USP30 (0.41) USP30PAX8CHRNB2CHRNA4NPC1
SCHEMBL7225292 0.86 P2RX7 (0.43) USP30SLC6A3AXLMERTKCHRNB2
SCHEMBL7224212 0.86 USP30 (0.41) USP30SLC6A3CHRNB2CHRNA4NPC1
SCHEMBL7226302 0.86 NPC1 (0.52) USP30CYP2D6CYP2C19CHRNB2CHRNA4
SCHEMBL7071274 0.85 USP30 (0.53) USP30CYP3A4CYP2D6CYP2C19SLC6A3
Hydrochloric Acid SCHEMBL7075524 0.84 USP30 (0.52) USP30CYP3A4CYP2D6CYP2C19SLC6A3
SCHEMBL7232527 0.84 USP30 (0.42) USP30SLC6A3HTR3ACHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed