SCHEMBL7233105

SCHEMBL7233105

O=C(Nc1ccc(-n2nc(C(F)(F)F)cc2C(F)(F)F)cc1)Nc1cc(Cl)cc(Cl)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ORAI1 Q96D31 3/20 0.70
TP53 P04637 2/20 0.61
MAPT P10636 5/20 0.58
THRB P10828 1/20 0.57
TRPC3 Q13507 3/20 0.56
TRPC1 P48995 1/20 0.56
STIM1 Q13586 1/20 0.56
TRPC5 Q9UL62 1/20 0.55
NPSR1 Q6W5P4 1/20 0.54
KCNJ6 P48051 2/20 0.51
KCNJ5 P48544 2/20 0.51
KCNJ3 P48549 2/20 0.51
NPC1 O15118 2/20 0.48
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
MAPK14 Q16539 1/20 0.47
RAB9A P51151 1/20 0.46
CRACR2A Q9BSW2 2/20 0.46
PTGS2 P35354 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7235013 0.87 TP53 (0.62) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7320311 0.86 ORAI1 (0.67) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7319407 0.86 TP53 (0.64) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7315526 0.86 TP53 (0.71) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7314472 0.86 TP53 (0.67) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7313426 0.83 ORAI1 (0.67) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7321880 0.82 ORAI1 (1.00) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL5208645 0.82 ORAI1 (1.00) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7325234 0.81 ORAI1 (0.67) ORAI1TP53MAPTTHRBTRPC3
SCHEMBL7322521 0.81 ORAI1 (0.58) ORAI1TP53MAPTTHRBTRPC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506747-B1 Method of treating an inflammatory disease which comprises administering to a patient in need of such treatment-a N-(4-(5-Ethyl-3-pyridin-3-yl-pyrazol-1-yl)phenyl)pyridine-3-carboxamide; BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2003-01-14 US disclosed