SCHEMBL7235686

SCHEMBL7235686

c1cnc2cc3cnccc3cc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 2/20 0.54
CSNK1D P48730 1/20 0.54
CSNK1E P49674 1/20 0.54
DYRK1A Q13627 1/20 0.54
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
POLB P06746 1/20 0.47
PDGFRB P09619 2/20 0.46
PDGFRA P16234 2/20 0.46
CASP6 P55212 1/20 0.44
ALDH1A1 P00352 5/20 0.44
CASP1 P29466 2/20 0.44
HTT P42858 2/20 0.44
MEN1 O00255 1/20 0.44
CASP7 P55210 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
NR4A2 P43354 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750534 1.00 CLK1 (0.54) CLK1CSNK1DCSNK1EDYRK1ANPC1
Isoquinoline SCHEMBL7993276 0.95 CLK1 (0.50) CLK1CSNK1DCSNK1EDYRK1ANPC1
Quinoline SCHEMBL7992158 0.93 ALDH1A1 (0.57) CLK1CSNK1DCSNK1EDYRK1ANPC1
SCHEMBL50867 0.83 ALDH1A1 (0.61) DYRK1ANPC1RAB9APOLBPDGFRB
SCHEMBL29726025 0.83 ALDH1A1 (0.61) DYRK1ANPC1RAB9APOLBPDGFRB
SCHEMBL31733917 0.81 ALDH1A1 (0.58) DYRK1ANPC1RAB9APOLBPDGFRB
SCHEMBL29471812 0.81 ALDH1A1 (0.58) DYRK1ANPC1RAB9APOLBPDGFRB
Ammonia Solution, Strong SCHEMBL29036762 0.81 ALDH1A1 (0.58) DYRK1ANPC1RAB9APOLBPDGFRB
SCHEMBL29845770 0.81 ALDH1A1 (0.58) DYRK1ANPC1RAB9APOLBPDGFRB
SCHEMBL30422685 0.81 ALDH1A1 (0.58) DYRK1ANPC1RAB9APOLBPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624933-A Process for the preparation of a 6-fluoro-2-halo-quinoline RHONE-POULENC RORER S.A. (FR) 1997-04-29 US claimed
JP-2300171-A None JP disclosed
JP-3056464-A None JP disclosed
US-20250073225-A1 BIFUNCTIONAL COMPOSITIONS FOR THE TREATMENT OF CANCER ARMACEUTICA INC (US) 2025-03-06 US disclosed
US-12201626-B2 Bifunctional compositions for the treatment of cancer Armaceutica, Inc. (US) 2025-01-21 US disclosed
EP-3793544-B1 BIFUNCTIONAL COMPOSITIONS FOR THE TREATMENT OF CANCER ARMACEUTICA INC (US) 2023-09-20 EP disclosed
US-20210361643-A1 BIFUNCTIONAL COMPOSITIONS FOR THE TREATMENT OF CANCER ARMACEUTICA INC (US) 2021-11-25 US disclosed
CN-112672741-A Bifunctional compositions for treating cancer 阿玛切蒂卡有限公司 2021-04-16 CN disclosed
EP-3793544-A1 BIFUNCTIONAL COMPOSITIONS FOR THE TREATMENT OF CANCER Armaceutica, Inc (US) 2021-03-24 EP disclosed
US-10862046-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2020-12-08 US disclosed
EP-0379412-B1 1,8-Benzonaphthyridine derivatives, their preparation and compositions containing them BELLON LABOR SA ROGER (FR) 1993-12-01 EP disclosed
EP-0536035-A1 1,8-Benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1993-04-07 EP disclosed
US-5091535-A ORGANIC PHOTOCHROMIC COMPOUND, A DIMER OF PYRIDO QUINOLINE SEIKISUI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1992-02-25 US disclosed
EP-0431991-A1 1,8-Benzonaphthyridine derivatives, their preparation and compositions containing them Société anonyme dite: LABORATOIRE ROGER BELLON (FR) 1991-06-12 EP disclosed
JP-H0356464-A 3-PYRIDYL-2-(3-METHYL PYRIDYL)METHANE AND PRODUCTION THEREOF SEKISUI CHEM CO LTD 1991-03-12 JP disclosed
JP-H02300171-A 3-PYRIDYL-2-(3-METHYLPYRIDYL)METHANOL AND PREPARATION THEREOF SEKISUI CHEM CO LTD 1990-12-12 JP disclosed
EP-0394846-A2 Organic photochromic compound SEKISUI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1990-10-31 EP disclosed
EP-0379414-A1 1,8-Benzonaphthyridine derivatives and their preparation Société anonyme dite: LABORATOIRE ROGER BELLON (FR) 1990-07-25 EP disclosed
EP-0379412-A1 1,8-Benzonaphthyridine derivatives, their preparation and compositions containing them Société anonyme dite: LABORATOIRE ROGER BELLON (FR) 1990-07-25 EP disclosed
EP-0379413-A1 1,8-Benzonaphthyridine derivatives, their production and compositions containing them Société anonyme dite: LABORATOIRE ROGER BELLON (FR) 1990-07-25 EP disclosed