Isoquinoline

Isoquinoline

SCHEMBL7993276

c1ccc2cnccc2c1.c1cnc2cc3cnccc3cc2c1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 2/20 0.50
CSNK1D P48730 1/20 0.50
CSNK1E P49674 1/20 0.50
DYRK1A Q13627 1/20 0.50
ALDH1A1 P00352 5/20 0.44
NPC1 O15118 2/20 0.44
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
CYP2A6 P11509 1/20 0.42
PDGFRB P09619 2/20 0.42
PDGFRA P16234 2/20 0.42
CYP17A1 P05093 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
MAPT P10636 2/20 0.42
CASP6 P55212 1/20 0.41
CASP1 P29466 2/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7235686 0.95 CLK1 (0.54) CLK1CSNK1DCSNK1EDYRK1AALDH1A1
SCHEMBL4750534 0.95 CLK1 (0.54) CLK1CSNK1DCSNK1EDYRK1AALDH1A1
Quinoline SCHEMBL7992158 0.92 ALDH1A1 (0.57) CLK1CSNK1DCSNK1EDYRK1AALDH1A1
SCHEMBL29726025 0.83 ALDH1A1 (0.61) DYRK1AALDH1A1NPC1POLBRAB9A
SCHEMBL50867 0.83 ALDH1A1 (0.61) DYRK1AALDH1A1NPC1POLBRAB9A
Anthracene SCHEMBL29011110 0.83 CYP19A1 (0.50) CLK1CSNK1DCSNK1EDYRK1APOLB
Isoquinoline SCHEMBL1505711 0.82 ALDH1A1 (0.68) CLK1ALDH1A1NPC1POLBRAB9A
Isoquinoline SCHEMBL27938240 0.82 ALDH1A1 (0.68) CLK1ALDH1A1NPC1POLBRAB9A
SCHEMBL29066655 0.81 ALDH1A1 (0.58) DYRK1AALDH1A1NPC1POLBRAB9A
SCHEMBL31733917 0.81 ALDH1A1 (0.58) DYRK1AALDH1A1NPC1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017997-A1 SUBSTITUTED DIAZAANTHRACENE COMPOUNDS HAVING PHARMACEUTICAL UTILITY DIAZANS LIMITED (CA) 2001-03-15 WO disclosed