SCHEMBL7236366

SCHEMBL7236366

O=C(O)C(O)=CC(=O)c1cnn(S(=O)(=O)c2ccc(Cl)cc2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 4/20 0.34
AKR1C3 P42330 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH3A1 P30838 2/20 0.34
CNR1 P21554 1/20 0.34
AKR1C2 P52895 1/20 0.34
AKR1C1 Q04828 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HSD11B1 P28845 1/20 0.34
LMNA P02545 2/20 0.33
PPARG P37231 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7236361 1.00 TSHR (0.35) TSHRMEN1KMT2AALDH1A1AKR1C3
SCHEMBL4675007 0.79 AKR1C3 (0.44) MEN1KMT2AALDH1A1AKR1C3KDM4E
SCHEMBL4674580 0.75 ALDH1A1 (0.39) MEN1KMT2AALDH1A1AKR1C3CNR1
SCHEMBL4673009 0.73 ALDH1A1 (0.45) MEN1KMT2AALDH1A1AKR1C3KDM4E
SCHEMBL4672360 0.69 RAPGEF4 (0.47) ALDH1A1AKR1C3KDM4EALDH3A1AKR1C2
SCHEMBL4677989 0.69 ALDH1A1 (0.63) MEN1KMT2AALDH1A1AKR1C3KDM4E
SCHEMBL4677987 0.69 ALDH1A1 (0.63) MEN1KMT2AALDH1A1AKR1C3KDM4E
SCHEMBL4672356 0.69 RAPGEF4 (0.47) ALDH1A1AKR1C3KDM4EALDH3A1AKR1C2
SCHEMBL4672259 0.68 ALDH1A1 (0.37) MEN1KMT2AALDH1A1AKR1C3AKR1C2
SCHEMBL4672257 0.68 ALDH1A1 (0.37) MEN1KMT2AALDH1A1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6645956-B1 1-(5-(4-fluorobenzyl)furan-2-yl)-3-hydroxy-3-(1H-1,2,4-triazol-3 -yl)-propenone; viricides; AIDS treatment SHIONOGI & CO., LTD. (JP) 2003-11-11 US disclosed