SCHEMBL7238041

SCHEMBL7238041

CCCCS(=O)(=O)NC(Cc1ccc(OCC2CN(CCN3CCN(C(=O)OC(C)(C)C)CC3)C(=O)O2)cc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.46
ITGA2B P08514 8/20 0.46
ITGAV P06756 1/20 0.46
CHRM2 P08172 1/20 0.46
SLC6A4 P31645 1/20 0.46
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
YAP1 P46937 2/20 0.41
MMP13 P45452 2/20 0.38
MMP2 P08253 1/20 0.38
HRH2 P25021 3/20 0.38
HRH1 P35367 3/20 0.38
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7237602 0.97 ITGB3 (0.47) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7237692 0.97 ITGB3 (0.47) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7238454 0.95 YAP1 (0.41) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7228601 0.91 MAPK1 (0.42) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7228442 0.91 MAPK1 (0.42) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7229936 0.86 YAP1 (0.48) ITGB3ITGA2BMAPK1L3MBTL1YAP1
SCHEMBL7228788 0.84 HRH2 (0.49) ITGB3ITGA2BMAPK1L3MBTL1YAP1
SCHEMBL7231440 0.84 HRH2 (0.49) ITGB3ITGA2BMAPK1L3MBTL1YAP1
SCHEMBL7228364 0.81 YAP1 (0.48) YAP1HRH2HRH1
SCHEMBL7235241 0.81 ITGB3 (0.44) ITGB3ITGA2BITGAVCHRM2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed