SCHEMBL7238595

SCHEMBL7238595

COC(=O)CCCc1c(-c2ccc(Br)cc2)[nH]c2ccc(Cl)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 3/20 0.53
TSPO P30536 1/20 0.49
TACR1 P25103 5/20 0.49
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
HPGD P15428 1/20 0.48
CYP2C19 P33261 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MC4R P32245 1/20 0.45
SIRT1 Q96EB6 1/20 0.43
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7238513 0.93 TSPO (0.56) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7241810 0.89 CXCR2 (0.56) CXCR2TSPOTACR1
SCHEMBL7242413 0.88 TSPO (0.46) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7241409 0.87 TSPO (0.47) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7232861 0.87 TSPO (0.47) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7790369 0.87 CXCR2 (0.52) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7233759 0.87 CXCR2 (0.52) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7241216 0.87 TACR1 (0.45) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7236310 0.87 TACR1 (0.49) CXCR2TSPOTACR1KDM4EALDH1A1
SCHEMBL7232319 0.87 CXCR2 (0.55) CXCR2TSPOTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6605633-B1 Such as 5-Bromo-2-phenyl-1H-indole-3-butanoic acid FOURNIER INDUSTRIE ET SANTE (FR) 2003-08-12 US disclosed
CN-1391556-A novel IL-8 receptor antagonists FOURNIER IND & SANTE (FR) 2003-01-15 CN disclosed