SCHEMBL7239483

SCHEMBL7239483

COc1ccc2c(c1)-c1nc(Nc3cc(O)c(OC)c(OC)c3)ncc1CS2

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.68
CA12 O43570 2/20 0.56
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
CA9 Q16790 2/20 0.56
EGFR P00533 2/20 0.55
PLK1 P53350 1/20 0.49
IKBKB O14920 1/20 0.46
FYN P06241 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997904 0.85 FYN (0.61) KDRPLK1IKBKBFYN
SCHEMBL7238828 0.84 KDR (0.65) KDRCA12CA1CA2CA9
SCHEMBL7241137 0.82 KDR (0.72) KDRCA12CA1CA2CA9
Hydrochloric Acid SCHEMBL7242637 0.80 FYN (0.59) KDRPLK1IKBKBFYN
SCHEMBL7237418 0.79 FYN (0.65) KDRPLK1IKBKBFYN
SCHEMBL7235444 0.77 IKBKB (0.67) KDRCA12CA1CA2CA9
Hydrochloric Acid SCHEMBL7516453 0.76 IKBKB (0.66) KDRCA12CA1CA2CA9
SCHEMBL7241237 0.76 KDR (0.66) KDRCA12CA1CA2CA9
SCHEMBL6998752 0.75 IKBKB (0.58) KDRCA12CA1CA2CA9
SCHEMBL6992464 0.75 KDR (0.65) KDRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599908-B1 Potent and selective inhibitors of the protein tyrosine kinases p56lck and p59fyn CELLTECH R & D LIMITED (GB) 2003-07-29 US disclosed
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed