SCHEMBL7242520

SCHEMBL7242520

Nc1cccc(OCCN2CCCCC2Cc2ccc(Cl)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SPHK2 Q9NRA0 5/20 0.47
SPHK1 Q9NYA1 5/20 0.47
LTA4H P09960 5/20 0.46
HRH3 Q9Y5N1 2/20 0.43
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7247786 0.95 SPHK2 (0.47) SPHK2SPHK1LTA4HHRH3
SCHEMBL7247863 0.90 LTA4H (0.48) SPHK2SPHK1LTA4HSMN1; SMN2
SCHEMBL7249762 0.84 KDM4E (0.46) SPHK2SPHK1LTA4HHRH3
SCHEMBL7244329 0.82 SIGMAR1 (0.47) SPHK2SPHK1HRH3
SCHEMBL7244055 0.80 LTA4H (0.50) LTA4HHRH3
SCHEMBL7251610 0.80 LTA4H (0.50) LTA4HHRH3
Hydrochloric Acid SCHEMBL7508739 0.79 LTA4H (0.49) LTA4HHRH3
Hydrochloric Acid SCHEMBL7246199 0.79 LTA4H (0.49) LTA4HHRH3
Hydrochloric Acid SCHEMBL7243161 0.79 LTA4H (0.49) LTA4HHRH3
SCHEMBL7400679 0.78 LTA4H (0.41) SPHK2SPHK1LTA4HHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534525-B1 Method of using 2- substituted piperidine analogs as selectively active antagonist of N-methyl-D-aspartate (NMDA) receptor subtypes for treating conditions such as stroke, cerebral ischemia, central nervous system trauma, WARNER-LAMBERT & COMPANY 2003-03-18 US disclosed
US-6124317-A ACTIVE DRUG TREATING STROKE, CEREBRAL ISCHEMIA, CENTRAL NERVOUS SYSTEM TRAUMA, HYPOGLYCEMIA, ANXIETY, CONVULSIONS, AMIOGLYCOSIDE ANTIBIOTICS-INDUCED HEARING LOSS, MIGRAINE HEADACHES, CHRONIC PAIN, GLAUCOMA, CMV RETINITIS, PSYCHOSIS WARNER-LAMBERT COMPANY (US) 2000-09-26 US disclosed