SCHEMBL7243165

SCHEMBL7243165

CNC(=O)c1cccc(NC(=O)COc2ccc3ccccc3c2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.60
KCNH2 Q12809 1/20 0.59
LMNA P02545 2/20 0.59
GALR3 O60755 1/20 0.59
STAT3 P40763 1/20 0.59
ALDH1A1 P00352 1/20 0.58
SIRT5 Q9NXA8 1/20 0.58
KMT2A Q03164 4/20 0.57
MEN1 O00255 3/20 0.57
RAB9A P51151 4/20 0.57
POLB P06746 3/20 0.57
NPC1 O15118 3/20 0.57
CASP3 P42574 1/20 0.57
SENP8 Q96LD8 1/20 0.57
SENP7 Q9BQF6 1/20 0.57
SENP6 Q9GZR1 1/20 0.57
CYP1A2 P05177 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7237041 0.88 MAPT (0.78) MAPTKCNH2LMNAALDH1A1KMT2A
SCHEMBL2958454 0.86 HIF1A (0.71) MAPTLMNAGALR3STAT3ALDH1A1
SCHEMBL7243115 0.83 KCNH2 (0.68) MAPTKCNH2LMNAALDH1A1KMT2A
SCHEMBL7239320 0.82 DAPK1 (0.77) MAPTKCNH2LMNAALDH1A1SIRT5
SCHEMBL4738194 0.82 GALR3 (0.79) MAPTLMNAGALR3STAT3ALDH1A1
SCHEMBL7168527 0.81 L3MBTL1 (0.69) MAPTLMNAALDH1A1SIRT5KMT2A
SCHEMBL7238805 0.80 RAB9A (0.78) MAPTLMNAALDH1A1KMT2AMEN1
SCHEMBL7244929 0.80 SMN1; SMN2 (0.64) MAPTALDH1A1KMT2AMEN1RAB9A
SCHEMBL25463130 0.79 RAB9A (0.72) LMNAGALR3STAT3ALDH1A1KMT2A
SCHEMBL2332894 0.79 GALR3 (0.66) LMNAGALR3STAT3KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030083523-A1 Amide derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2003-05-01 US claimed
EP-0887341-A1 Amide derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 1998-12-30 EP claimed
US-20030083523-A1 Amide derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2003-05-01 US disclosed
US-6444849-B1 BACTERICIDES MITSUBISHI CHEMICAL CORPORATION (JP) 2002-09-03 US disclosed
EP-0887341-A1 Amide derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 1998-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030083523-A1 Amide derivatives H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CBR3, CBR1 MAPT 3965/4885KCNH2 228/4885LMNA 1674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.