SCHEMBL7245239

SCHEMBL7245239

COc1cc(C(=O)C(=O)N2CC[C@H]2C(=O)O)cc(OC)c1OC

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 14/20 0.66
MMP2 P08253 1/20 0.48
ANPEP P15144 1/20 0.48
GAA P10253 1/20 0.47
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
ABCC1 P33527 1/20 0.44
FKBP4 Q02790 1/20 0.44
FKBP5 Q13451 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1233422 0.92 FKBP1A (0.74) FKBP1AMMP2ANPEPABCC1FKBP4
SCHEMBL1233420 0.92 FKBP1A (0.74) FKBP1AMMP2ANPEPABCC1FKBP4
SCHEMBL5966161 0.91 FKBP1A (0.80) FKBP1AABCC1FKBP4FKBP5
SCHEMBL7155851 0.91 FKBP1A (0.80) FKBP1AABCC1FKBP4FKBP5
Hydroxyamine SCHEMBL5274861 0.84 GAA (0.53) FKBP1AMMP2ANPEPGAAALDH1A1
Hydroxyamine SCHEMBL5274854 0.84 GAA (0.53) FKBP1AMMP2ANPEPGAAALDH1A1
SCHEMBL14407836 0.79 FKBP1A (0.63) FKBP1AMMP2ANPEPGAAALDH1A1
SCHEMBL5966113 0.79 FKBP1A (0.63) FKBP1AMMP2ANPEPALDH1A1FKBP5
SCHEMBL11998537 0.78 FKBP1A (0.56) FKBP1AMMP2ANPEPGAAALDH1A1
SCHEMBL1233000 0.77 FKBP1A (0.73) FKBP1AABCC1FKBP4FKBP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6544976-B1 Treating disorders characterized by neuronal damage caused by disease or trauma, such as Parkinson's disease, Alzheimer's disease, stroke, multiple sclerosis, amyotrophic lateral sclerosis, diabetic neuropathy and Bell's palsy. ORTHO-MCNEIL PHARMACEUTICAL, INC. 2003-04-08 US disclosed
WO-2001004091-A1 NEUROTROPHIC 2-AZETIDINECARBOXYLIC ACID DERIVATIVES, AND RELATED COMPOSITIONS AND METHODS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-01-18 WO disclosed