SCHEMBL7248276

SCHEMBL7248276

[CH2]N(Cc1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
ALDH1A1 P00352 3/20 0.48
AOC3 Q16853 1/20 0.44
CYP2C19 P33261 1/20 0.43
NPC1 O15118 1/20 0.42
GLA P06280 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
PAX8 Q06710 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CNR2 P34972 1/20 0.41
CA2 P00918 1/20 0.40
MAOB P27338 1/20 0.40
CALM1 P0DP23 1/20 0.39
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
MGLL Q99685 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1776018 0.76 TSHR (0.55) TSHRALDH1A1AOC3CYP2C19NPC1
SCHEMBL5462064 0.76 TSHR (0.55) TSHRALDH1A1AOC3CYP2C19NPC1
SCHEMBL11512451 0.75 TSHR (0.50) TSHRALDH1A1AOC3CYP2C19NPC1
Ethylene SCHEMBL11428459 0.75 NR3C2 (0.53) TSHRALDH1A1AOC3CYP2C19NPC1
SCHEMBL918512 0.74 NR3C2 (0.56) TSHRALDH1A1AOC3CYP2C19NPC1
SCHEMBL43183 0.74 TSHR (0.74) TSHRALDH1A1AOC3CYP2C19GLA
Hydrochloric Acid SCHEMBL2139953 0.72 TSHR (0.71) TSHRALDH1A1AOC3CYP2C19GLA
SCHEMBL10842660 0.72 TSHR (0.50) TSHRALDH1A1AOC3CYP2C19NPC1
SCHEMBL94987 0.72 TSHR (0.46) TSHRALDH1A1CYP2C19GLAHTT
SCHEMBL294642 0.72 TSHR (0.64) TSHRALDH1A1AOC3CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0039903-B1 8-SUBSTITUTED PYRROLIZIDINES AND QUATERNARY AMMONIUM SALTS THEREOF SUNTORY KABUSHIKI KAISHA (JP) 1986-04-09 EP claimed
US-6514988-B1 A pregnancy controlling agent and a menstrual cycle controlling agent; useful as an agent of spawning promotion in fish TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-04 US disclosed
CN-1092197-C Bicyclic thiophene derivatives and use as gonadotropin releasing hormone antagonists TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-09 CN disclosed
US-6187788-B1 THIENO(2,3-B)(DIHYDRO)PYRIDINE DERIVATIVES; GONADOTROPIN-RELEASING HORMONE ANTAGONISTS; ANTICARCINOGENIC AGENTS; SEXUAL AND UROGENITAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-02-13 US disclosed
CN-1146206-A Bicyclic thiophene derivatives and use as gonadotropin releasing hormone antagonists TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-03-26 CN disclosed
EP-0039903-B1 8-SUBSTITUTED PYRROLIZIDINES AND QUATERNARY AMMONIUM SALTS THEREOF SUNTORY KABUSHIKI KAISHA (JP) 1986-04-09 EP disclosed