SCHEMBL724850

SCHEMBL724850

C=CCc1ccc(OC(=O)C(CCC)CCC)c(-c2cc(CC=C)ccc2OC(CCNC)c2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 6/20 0.44
SLC6A4 P31645 14/20 0.42
SLC6A2 P23975 10/20 0.42
CYP2D6 P10635 8/20 0.42
CYP1A2 P05177 4/20 0.42
CYP3A4 P08684 4/20 0.42
KCNH2 Q12809 4/20 0.42
TSHR P16473 3/20 0.42
SLC6A3 Q01959 3/20 0.42
KMT2A Q03164 2/20 0.42
CHRM1 P11229 2/20 0.42
ADRA2B P18089 2/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HRH1 P35367 2/20 0.42
OPRM1 P35372 2/20 0.42
DRD3 P35462 2/20 0.42
OPRK1 P41145 2/20 0.42
HTR2B P41595 2/20 0.42
KLF10 Q13118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL530776 0.99 NOS2 (0.44) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
Hydrochloric Acid SCHEMBL726040 0.91 NOS2 (0.40) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
SCHEMBL526595 0.85 NOS2 (0.47) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
SCHEMBL526594 0.85 NOS2 (0.47) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
Hydrochloric Acid SCHEMBL726039 0.84 NOS2 (0.40) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
SCHEMBL525534 0.83 GABRA1 (0.54) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
SCHEMBL525899 0.83 SLC6A4 (0.52) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
SCHEMBL525549 0.83 SLC6A4 (0.59) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
Hydrochloric Acid SCHEMBL726060 0.82 SLC6A4 (0.51) NOS2SLC6A4SLC6A2CYP2D6CYP1A2
Hydrochloric Acid SCHEMBL530274 0.82 GABRA1 (0.53) NOS2SLC6A4SLC6A2CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP claimed
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO disclosed