SCHEMBL7248696

SCHEMBL7248696

CS(=O)(=O)NCC1(CN)CCN(Cc2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ALDH1A1 P00352 2/20 0.45
NPFFR1 Q9GZQ6 5/20 0.45
NPFFR2 Q9Y5X5 5/20 0.45
OPRK1 P41145 1/20 0.45
CYP3A4 P08684 3/20 0.44
TSHR P16473 2/20 0.44
HSD17B10 Q99714 1/20 0.44
OPRL1 P41146 2/20 0.43
SIGMAR1 Q99720 1/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
HIF1A Q16665 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254428 0.84 CNR2 (0.52) CYP2D6ALDH1A1NPFFR1NPFFR2OPRK1
SCHEMBL3334062 0.80 SIGMAR1 (0.61) CYP2D6MEN1KMT2AALDH1A1CYP3A4
SCHEMBL7251032 0.80 NPFFR1 (0.56) CYP2D6ALDH1A1NPFFR1NPFFR2OPRK1
SCHEMBL6887496 0.79 CYP2D6 (0.48) CYP2D6MEN1KMT2AALDH1A1NPFFR1
SCHEMBL7253609 0.79 CYP3A4 (0.49) CYP2D6MEN1KMT2AALDH1A1CYP3A4
SCHEMBL2277424 0.78 CYP2D6 (0.51) CYP2D6MEN1KMT2AALDH1A1CYP3A4
SCHEMBL20571382 0.78 CYP3A4 (0.54) CYP2D6MEN1KMT2AALDH1A1NPFFR1
SCHEMBL7249627 0.77 MAPK1 (0.50) CYP2D6MEN1KMT2AALDH1A1NPFFR1
SCHEMBL4630842 0.76 POLB (0.57) MEN1KMT2AALDH1A1NPFFR1NPFFR2
SCHEMBL7248229 0.76 NPFFR1 (0.60) NPFFR1NPFFR2OPRK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545022-B1 Treatment of epilepsy, faintness attacks, hypokinesia, cranial disorders, neurodegenerative disorders, depression, anxiety, panic, pain, neuropathological disorders, inflammatory diseases, and gastrointestinal disorders PFIZER INC. 2003-04-08 US disclosed