SCHEMBL7248756

SCHEMBL7248756

O=C(NO)C1(CS(=O)(=O)N2CCN(c3ccc(Cl)cc3)CC2)CCC2(CC1)OCCO2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 7/20 0.52
MMP9 P14780 7/20 0.52
MMP13 P45452 6/20 0.52
MMP3 P08254 3/20 0.52
MMP14 P50281 3/20 0.52
MMP8 P22894 2/20 0.52
MMP1 P03956 2/20 0.50
ADAM10 O14672 2/20 0.50
ABCB11 O95342 1/20 0.45
MMP7 P09237 1/20 0.45
MMP10 P09238 1/20 0.45
ADAM17 P78536 1/20 0.45
POLB P06746 2/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALDH1A1 P00352 2/20 0.41
ADAMTS4 O75173 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12152323 0.89 MMP2 (0.61) MMP2MMP9MMP13MMP3MMP14
SCHEMBL7249415 0.89 POLB (0.44) MMP2MMP9MMP13MMP3MMP14
SCHEMBL7248141 0.84 MMP2 (0.49) MMP2MMP9MMP13MMP3MMP14
SCHEMBL7249713 0.83 MAPT (0.46) MMP2MMP9MMP13MMP3MMP14
SCHEMBL6782627 0.80 MMP2 (0.56) MMP2MMP9MMP13MMP3MMP14
SCHEMBL4816291 0.79 ADAMTS4 (0.60) MMP2MMP9MMP13MMP3MMP14
SCHEMBL7255900 0.79 MMP2 (0.46) MMP2MMP9MMP13MMP3MMP14
SCHEMBL6785924 0.73 MMP2 (0.52) MMP2MMP9MMP13MMP3MMP14
SCHEMBL6787148 0.73 MMP2 (0.51) MMP2MMP9MMP13MMP3MMP14
SCHEMBL6950652 0.72 MMP2 (0.58) MMP2MMP9MMP13MMP3MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6503910-B1 Metalloproteinase inhibitors; antimetastasis agents; arthritis, neurodegenerative disorder treatment DARWIN DISCOVERY LTD. (GB) 2003-01-07 US claimed
EP-1177183-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES Darwin Discovery Limited (GB) 2002-02-06 EP claimed
WO-2000069839-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES DARWIN DISCOVERY LIMITED (GB) 2000-11-23 WO claimed