SCHEMBL7248995

SCHEMBL7248995

CCS(=O)(=O)Nc1cc(Cc2c[nH]cn2)c(C)cc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.40
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HPGD P15428 2/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
JAK2 O60674 3/20 0.32
JAK1 P23458 3/20 0.32
TYK2 P29597 3/20 0.32
JAK3 P52333 3/20 0.32
PDE10A Q9Y233 1/20 0.32
TP53 P04637 1/20 0.32
LMNA P02545 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP2C9 P11712 1/20 0.31
PSIP1 O75475 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
ADRA2A P08913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7097637 0.81 BRD4 (0.32) BRD4HTTHPGDPDE10ALMNA
SCHEMBL7102580 0.81 HPGD (0.40) BRD4HTTSMN1; SMN2HPGDJAK2
SCHEMBL7105179 0.81 HPGD (0.39) BRD4HTTSMN1; SMN2HPGDKDM4E
SCHEMBL7248476 0.79 BRAF (0.34) HTTHPGDJAK2JAK1TYK2
SCHEMBL7103450 0.79 BRD4 (0.31) BRD4HTTPDE10A
SCHEMBL7248382 0.79 NR3C1 (0.41) HTTSMN1; SMN2HPGDALDH1A1PDE10A
SCHEMBL7103402 0.78 MRGPRX1 (0.34) HTTJAK2JAK1TYK2JAK3
SCHEMBL7254139 0.76 HPGD (0.31) HTTSMN1; SMN2HPGDLMNA
SCHEMBL7249546 0.76 HPGD (0.33) BRD4HTTSMN1; SMN2HPGDKDM4E
SCHEMBL7248262 0.76 MEN1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6503935-B1 Treating urinary incontinence or retrograde ejaculation ABBOTT LABORATORIES 2003-01-07 US disclosed
EP-1102754-A1 IMIDAZOLES AND RELATED COMPOUNDS AS ALPHA-1A AGONISTS ABBOTT LABORATORIES (US) 2001-05-30 EP disclosed
WO-2000007997-A1 IMIDAZOLES AND RELATED COMPOUNDS AS α1A AGONISTS ABBOTT LABORATORIES (US) 2000-02-17 WO disclosed