SCHEMBL7250707

SCHEMBL7250707

COc1nc([NH])nc(N)n1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1576395 0.82 TSHR (0.44) TP53POLBGAATSHRHTT
SCHEMBL138352 0.82 HSD17B10 (0.44) TP53POLBGAATSHRHTT
SCHEMBL441545 0.73 HSP90AB1 (0.43) TP53POLBGAATSHRHTT
SCHEMBL30562916 0.73 HSP90AB1 (0.43) TP53POLBGAATSHRHTT
SCHEMBL2871435 0.73
SCHEMBL9190048 0.71 CYP1A2 (0.44) TSHR
SCHEMBL1577050 0.71 HSP90AA1 (0.50) TP53POLBGAATSHRHTT
SCHEMBL9266759 0.71 TP53 (0.39) TP53POLBGAATSHRHTT
Fluoride SCHEMBL31379739 0.71 HSP90AB1 (0.41) TP53POLBGAATSHRHTT
SCHEMBL10351075 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562844-B2 Attaching an olefin to a solid support; oxidizing the olefin to provide an epoxide functionality; opening the epoxide with an amine to form an amino alcohol; cyclizing the amino alcohol using a phosgene equivalent PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed