SCHEMBL7252243

SCHEMBL7252243

COc1cc(C)nc(OC(C(=O)O)C(OC=CCc2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 19/20 0.70
EDNRA P25101 19/20 0.70
NR1I2 O75469 1/20 0.58
KCNE1 P15382 1/20 0.58
KCNQ1 P51787 1/20 0.58
POLB P06746 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246331 0.92 EDNRB (0.66) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL7934042 0.83 EDNRB (1.00) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL7252235 0.82 EDNRB (0.89) EDNRBEDNRAPOLB
SCHEMBL7245599 0.80 EDNRB (0.80) EDNRBEDNRA
SCHEMBL6561931 0.79 EDNRB (0.77) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL795626 0.79 EDNRB (0.77) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL7252240 0.79 EDNRB (0.78) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL6561863 0.78 EDNRB (0.74) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL7245146 0.77 EDNRB (0.88) EDNRBEDNRA
SCHEMBL7252229 0.77 EDNRB (1.00) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6670367-B1 Vasodilator; hypertension; surprisingly show antagonistic action on the neurokinin receptor; 2-(4-Methoxy-6-methyl-2-pyrimidinyloxy)-3-(2-(3,4- dimethoxyphenyl)ethoxy)-3,3-diphenylpropionic Acid ABBOTT GMBH & CO., KG (DE) 2003-12-30 US disclosed