SCHEMBL7252899

SCHEMBL7252899

COC(=O)c1cc(N)c(SC)s1.CSc1sc(C(=O)O)c(C)c1NC(N)=S

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.33
OPRD1 P41143 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
CISD2 Q8N5K1 2/20 0.32
ALDH1A1 P00352 1/20 0.32
GRM6 O15303 1/20 0.31
GRM5 P41594 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
CASP3 P42574 1/20 0.30
RAB9A P51151 1/20 0.30
SENP8 Q96LD8 1/20 0.30
SENP7 Q9BQF6 1/20 0.30
SENP6 Q9GZR1 1/20 0.30
IKBKB O14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5839757 0.78 KEAP1 (0.41) GAAOPRD1KEAP1NFE2L2ALDH1A1
SCHEMBL6920646 0.73 ALDH1A1 (0.40) OPRD1KEAP1NFE2L2ALDH1A1KDM4E
SCHEMBL7836963 0.71 KEAP1 (0.57) KEAP1NFE2L2ALDH1A1KDM4EMAPT
SCHEMBL6921023 0.68 CSNK2A2 (0.38) GAAOPRD1KEAP1NFE2L2CISD2
SCHEMBL7983631 0.66 ALDH1A1 (0.33) OPRD1KEAP1NFE2L2ALDH1A1KDM4E
SCHEMBL6925163 0.66 KEAP1 (0.47) GAAOPRD1KEAP1NFE2L2ALDH1A1
SCHEMBL6921024 0.63 HPGD (0.39) GAAOPRD1KEAP1NFE2L2ALDH1A1
SCHEMBL6926946 0.62 KMT2A (0.52) GAACISD2NPC1MAPTRAB9A
SCHEMBL1417353 0.62 CSNK2A2 (0.45) GAAOPRD1ALDH1A1KDM4ENPC1
SCHEMBL3239031 0.62 KDM4E (0.54) GAAOPRD1ALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562840-B1 Non-peptidic inhibitors of proteolytic enzymes such as urokinase 3-DIMENSIONAL PHARMACEUTICALS, INC. 2003-05-13 US disclosed