SCHEMBL7253990

SCHEMBL7253990

Brc1ccc(-c2cnccc2C2CCCCC2)s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.37
RPS6KA3 P51812 2/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
OPRL1 P41146 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
CACNA1B Q00975 2/20 0.33
MAPT P10636 1/20 0.32
GSK3B P49841 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HSP90AA1 P07900 1/20 0.32
CYP17A1 P05093 3/20 0.32
CYP1A2 P05177 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7253763 0.93 RPS6KA3 (0.37) CYP11B2RPS6KA3MEN1KMT2AOPRL1
SCHEMBL7259043 0.82 CYP1A2 (0.48) CYP11B2RPS6KA3MEN1KMT2AOPRL1
SCHEMBL7257184 0.79 CYP1A2 (0.51) CYP11B2OPRL1SMN1; SMN2LMNAHPGD
SCHEMBL7258682 0.79 GCGR (0.45) CYP11B2RPS6KA3NPC1RAB9ASMN1; SMN2
SCHEMBL7257178 0.76 CYP3A4 (0.47) RPS6KA3NPC1RAB9ARXFP1MAPT
SCHEMBL7257212 0.76 APP (0.48) CYP11B2RPS6KA3CACNA1BHPGDALDH1A1
SCHEMBL7258670 0.74 CYP1A2 (0.51) CYP11B2RPS6KA3OPRL1CYP17A1CYP1A2
SCHEMBL7259298 0.73 CYP11B2 (0.47) CYP11B2OPRL1MAPTGSK3BALDH1A1
SCHEMBL7259545 0.72 CYP2A6 (0.47) RPS6KA3ALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL13735438 0.71 CYP11B2 (0.44) CYP11B2RPS6KA3OPRL1MAPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003027105-A1 SUBSTITUTED 3-PYRIDYL THIOPHENES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed