SCHEMBL7259043

SCHEMBL7259043

Cc1ccncc1-c1ccc(-c2cnccc2C2CCCCC2)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2E1 P05181 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C8 P10632 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2B6 P20813 1/20 0.48
CYP2C19 P33261 1/20 0.48
OPRL1 P41146 1/20 0.41
CYP11B2 P19099 4/20 0.36
ABL1 P00519 5/20 0.35
CYP11B1 P15538 3/20 0.34
RPS6KA3 P51812 2/20 0.34
CYP17A1 P05093 3/20 0.34
KIT P10721 1/20 0.34
PDGFRA P16234 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258670 0.93 CYP1A2 (0.51) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL7257184 0.83 CYP1A2 (0.51) CYP1A2CYP2E1CYP2C8CYP2D6CYP2A6
SCHEMBL7253990 0.82 CYP11B2 (0.37) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL7258682 0.80 GCGR (0.45) CYP2A6CYP11B2CYP11B1RPS6KA3CYP17A1
SCHEMBL7257178 0.80 CYP3A4 (0.47) CYP3A4CYP2A6CYP2C9CYP2C19RPS6KA3
SCHEMBL7257212 0.80 APP (0.48) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL7257157 0.78 CACNA1B (0.39) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL21757505 0.75 OPRL1 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL21757521 0.75 OPRL1 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7257202 0.75 CYP1A2 (0.54) CYP1A2CYP2E1CYP2C8CYP2D6CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003027105-A1 SUBSTITUTED 3-PYRIDYL THIOPHENES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed