SCHEMBL725522

SCHEMBL725522

CC(=O)OC=C(N)c1cc(C)c(Br)cc1O

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 1/20 0.31
PKM P14618 1/20 0.31
CYP1A1 P04798 1/20 0.30
CYP1B1 Q16678 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29836030 0.73 HTT (0.47) GRM1
SCHEMBL168765 0.73 HTT (0.47) GRM1
SCHEMBL722831 0.73 CASP3 (0.37) PKM
SCHEMBL722830 0.73 CASP3 (0.37) PKM
SCHEMBL167694 0.70 GRM1 (0.51) GRM1PKM
SCHEMBL168426 0.69 CA1 (0.50)
SCHEMBL11866432 0.69 ALDH1A1 (0.38) GRM1
SCHEMBL4261356 0.67 HTT (0.47)
SCHEMBL30922272 0.66 ALDH1A1 (0.39) GRM1
SCHEMBL26606973 0.65 ALDH1A1 (0.33) GRM1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609095-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2013-07-03 EP disclosed
EP-2563776-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2013-03-06 EP disclosed
WO-2012027710-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2012-03-01 WO disclosed
WO-2011139489-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-11-10 WO disclosed