SCHEMBL7255652

SCHEMBL7255652

CC(=O)Cc1ccc(CNc2nc(NCc3cccs3)nc3ccc(Cl)cc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.55
HRH1 P35367 1/20 0.55
HTR3A P46098 2/20 0.46
NPC1 O15118 1/20 0.46
CTNNB1 P35222 8/20 0.45
TCF7L2 Q9NQB0 8/20 0.45
CLK4 Q9HAZ1 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258507 0.89 HRH4 (0.55) HRH4HRH1HTR3ANPC1CTNNB1
SCHEMBL7260290 0.84 HRH4 (0.54) HRH4HRH1HTR3ANPC1CLK4
SCHEMBL7259297 0.83 HRH1 (0.50) HRH4HRH1CTNNB1TCF7L2
SCHEMBL7254578 0.83 HRH4 (0.60) HRH4HRH1HTR3ANPC1CLK4
SCHEMBL7258098 0.81 HRH1 (0.47) HRH4HRH1NPC1CTNNB1TCF7L2
SCHEMBL7254519 0.80 NPC1 (0.52) HRH4HRH1NPC1CTNNB1TCF7L2
SCHEMBL7259508 0.78 HRH4 (0.52) HRH4HRH1HTR3ANPC1CLK4
SCHEMBL2590769 0.75 RAD52 (0.68) HRH4HTR3A
SCHEMBL7254511 0.75 LMNA (0.56) CTNNB1TCF7L2CLK4
SCHEMBL21686898 0.71 HRH4 (1.00) HRH4HRH1HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055866-A1 QUINAZOLINE AND QUINOLINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO disclosed