SCHEMBL7255671

SCHEMBL7255671

Nc1n[nH]c2nc(-c3ccccc3)ncc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.49
GSK3A P49840 3/20 0.46
GSK3B P49841 3/20 0.46
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
RECQL P46063 1/20 0.46
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
JAK2 O60674 2/20 0.42
MAP4K4 O95819 1/20 0.42
CSF1R P07333 1/20 0.42
FGFR1 P11362 1/20 0.42
PDGFRA P16234 1/20 0.42
LTK P29376 1/20 0.42
KDR P35968 1/20 0.42
MAPK8 P45983 1/20 0.42
CSNK1A1 P48729 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16052176 0.78 MAPT (0.47) NPC1RAB9ALMNAMAPTKMT2A
SCHEMBL3174451 0.77 ADORA3 (0.48) LMNAKMT2APOLBADORA3ADORA2A
SCHEMBL3716787 0.75 NPC1 (0.46) NPC1RAB9ASMN1; SMN2LMNANR1H2
SCHEMBL23853930 0.74 GAA (0.53) GSK3AGSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL30675639 0.72 AURKB (0.51) GSK3AGSK3BRAB9AJAK2MAP4K4
SCHEMBL13329926 0.72 AURKB (0.51) GSK3AGSK3BRAB9AJAK2MAP4K4
SCHEMBL4697304 0.72 RET (0.41) GSK3AGSK3BKDRAURKBADORA2A
SCHEMBL30822335 0.72 RET (0.41) GSK3AGSK3BKDRAURKBADORA2A
SCHEMBL3762000 0.72 HPGDS (0.47) HPGDSGSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL5387619 0.71 GSK3B (0.59) GSK3AGSK3BJAK2MAP4K4CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8076338-B2 Such as 6-(4-phenylpiperazin-1-yl)-9H-purine; cell proliferation/differentiation EXELIXIS, INC. (US) 2011-12-13 US disclosed
WO-2003080617-A1 PYRAZOLOPYRIMIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-10-02 WO disclosed