SCHEMBL7255778

SCHEMBL7255778

C[C@H](CO)c1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 1/20 0.43
TRPA1 O75762 4/20 0.42
ABCB11 O95342 1/20 0.40
GAA P10253 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
CYP19A1 P11511 3/20 0.39
CYP17A1 P05093 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7255781 1.00 CYP3A4 (0.43) CYP3A4CYP2C19TRPA1ABCB11GAA
SCHEMBL11094130 0.82 TRPA1 (0.46) CYP3A4CYP2C19TRPA1GAASLC6A2
SCHEMBL2641075 0.82 ABCB11 (0.52) TRPA1ABCB11
SCHEMBL10031596 0.78 CYP3A4 (0.44) CYP3A4CYP2C19GAASLC6A2SLC6A4
SCHEMBL117057 0.78 CYP3A4 (0.44) CYP3A4CYP2C19GAASLC6A2SLC6A4
SCHEMBL17469429 0.78 CYP3A4 (0.44) CYP3A4CYP2C19GAASLC6A2SLC6A4
SCHEMBL21786012 0.77 CYP3A4 (0.40) CYP3A4CYP2C19TRPA1GAASLC6A2
SCHEMBL23689572 0.76 CYP3A4 (0.43) CYP3A4CYP2C19TRPA1GAASLC6A2
SCHEMBL21880656 0.76 CYP3A4 (0.43) CYP3A4CYP2C19GAASLC6A2SLC6A4
SCHEMBL11728032 0.76 TAAR1 (0.60) CYP3A4CYP2C19GAASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003006462-A1 PROCESSES FOR THE MANUFACTURE OF THROMBIN INHIBITORS AND N-PYRIDIN-4-YL-OXAZOLIDIN-2-ONES AS INTERMEDIATE THEREFOR GLAXO GROUP LIMITED (GB) 2003-01-23 WO disclosed