SCHEMBL7255877

SCHEMBL7255877

CC1CCC(NC(=O)c2cnc3cc4c(cc3n2)OCO4)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.56
RAB9A P51151 8/20 0.56
KMT2A Q03164 1/20 0.56
HPGDS O60760 1/20 0.47
KDM4E B2RXH2 2/20 0.42
MAPK1 P28482 2/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 1/20 0.41
CD38 P28907 1/20 0.41
HPGD P15428 2/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
CASP1 P29466 1/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TP53 P04637 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6083926 1.00 NPC1 (0.56) NPC1RAB9AKMT2AHPGDSKDM4E
SCHEMBL6084961 0.83 NPC1 (0.62) NPC1RAB9AKMT2AHPGDSLMNA
SCHEMBL7508967 0.83 NPC1 (0.62) NPC1RAB9AKMT2AHPGDSLMNA
SCHEMBL6083629 0.79 RAB9A (0.53) NPC1RAB9AHPGDSHPGDALDH1A1
SCHEMBL6085524 0.79 RAB9A (0.53) NPC1RAB9AHPGDSHPGDALDH1A1
SCHEMBL6083620 0.79 RAB9A (0.53) NPC1RAB9AHPGDSHPGDALDH1A1
SCHEMBL6085336 0.79 HPGDS (0.55) NPC1RAB9AKMT2AHPGDSLMNA
SCHEMBL6085327 0.79 HPGDS (0.55) NPC1RAB9AKMT2AHPGDSLMNA
SCHEMBL6085438 0.77 RAB9A (0.52) NPC1RAB9AKMT2AKDM4EMAPK1
SCHEMBL6085244 0.77 HPGDS (0.77) HPGDSCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500480-A 2003-01-07 JP claimed
EP-1196397-A1 METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS AND THEIR USE FOR TREATING CENTRAL NERVOUS SYSTEM DISEASES NPS PHARMACEUTICALS, INC. (US) 2002-04-17 EP claimed
WO-2000073283-A1 METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS AND THEIR USE FOR TREATING CENTRAL NERVOUS SYSTEM DISEASES NPS PHARMACEUTICALS, INC. (US) 2000-12-07 WO claimed