SCHEMBL7256357

SCHEMBL7256357

COC(=O)C(Cc1ccc(NC(=O)OC(C)(C)C)nc1)c1cn(CC(=O)C(C)(C)C)cn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 7/20 0.41
CPB1 P15086 8/20 0.39
NAMPT P43490 1/20 0.39
CPA1 P15085 2/20 0.38
GRIN2B Q13224 1/20 0.37
HDAC1 Q13547 1/20 0.37
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
HDAC3 O15379 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
SCD O00767 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7256257 0.87 NAMPT (0.43) CPB2CPB1NAMPTCPA1GRIN2B
SCHEMBL5465881 0.81 CPB1 (0.47) CPB2CPB1NAMPTCPA1GRIN2B
SCHEMBL5150256 0.79 NAMPT (0.46) CPB2NAMPTCPA1GRIN2BHDAC1
SCHEMBL5166294 0.78 NAMPT (0.40) CPB2NAMPTGRIN2BHDAC1GSK3B
SCHEMBL7257280 0.77 NAMPT (0.46) NAMPTGRIN2BHDAC1GSK3BDYRK1A
SCHEMBL7260251 0.76 CPB1 (0.51) CPB2CPB1NAMPTCPA1
SCHEMBL7260124 0.75 NAMPT (0.44) CPB2NAMPTGRIN2BHDAC1GSK3B
SCHEMBL7257206 0.75 CPB1 (0.46) CPB2CPB1CPA1GRIN2B
SCHEMBL12610053 0.74 CPB1 (0.52) CPB2CPB1NAMPTCPA1GRIN2B
SCHEMBL31407652 0.74 KLK5 (0.48) NAMPTGRIN2BHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003013526-A1 ANTICOAGULANT COMPOUNDS MERCK & CO. INC. (US) 2003-02-20 WO disclosed