SCHEMBL7257136

SCHEMBL7257136

O=C1CCn2c(N3CCC(O)CC3)nc3cccc1c32

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.37
OPRD1 P41143 3/20 0.37
OPRK1 P41145 3/20 0.37
OGFRL1 Q5TC84 3/20 0.37
PIK3CA P42336 2/20 0.37
PARP1 P09874 7/20 0.36
KCNH2 Q12809 4/20 0.35
GRM2 Q14416 4/20 0.35
PTPN11 Q06124 1/20 0.34
HTR3A P46098 2/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7257222 0.86 CCNE2 (0.39) OPRM1OPRD1OPRK1OGFRL1PIK3CA
SCHEMBL7257414 0.85 KCNH2 (0.39) PARP1KCNH2GRM2HTR3A
SCHEMBL7257413 0.85 PARP1 (0.36) PIK3CAPARP1KCNH2GRM2HTR3A
SCHEMBL6508880 0.84 CCR4 (0.39) OPRM1OPRD1OPRK1OGFRL1PARP1
SCHEMBL6633308 0.84 HRH1 (0.43) PARP1KCNH2GRM2PTPN11HTR3A
SCHEMBL7257145 0.82 KCNH2 (0.37) PARP1KCNH2GRM2HTR3AACHE
SCHEMBL6630805 0.82 PARP1 (0.43) PARP1HTR3A
SCHEMBL6631361 0.82 HDAC6 (0.46) PARP1KCNH2GRM2
SCHEMBL7262852 0.82 MAPK1 (0.33) PARP1KCNH2GRM2HTR3A
Hydrochloric Acid SCHEMBL6510200 0.81 PARP1 (0.42) PARP1HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003104233-A1 4,5-DIHYDRO-IMIDAZO (4,5,1-IJ) QUINOLIN-6-ONES DERIVATIVES AND THEIR USE AS POLY (ADP-RIBOSYL) TRANSFERASE (PARP) INHIBITORS ALTANA PHARMA AG (DE) 2003-12-18 WO disclosed