SCHEMBL6633308

SCHEMBL6633308

CN(C)C1CCN(c2nc3cccc4c3n2CCC4=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 8/20 0.43
KCNH2 Q12809 6/20 0.43
CYP2D6 P10635 5/20 0.43
CHEK2 O96017 1/20 0.38
PTPN11 Q06124 1/20 0.38
PARP1 P09874 5/20 0.37
CHRM1 P11229 3/20 0.36
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
MAOB P27338 1/20 0.34
HTR6 P50406 1/20 0.34
GRM2 Q14416 1/20 0.34
HTR3A P46098 1/20 0.34
CRHR1 P34998 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7257136 0.84 OPRM1 (0.37) KCNH2PTPN11PARP1GRM2HTR3A
SCHEMBL7257145 0.82 KCNH2 (0.37) KCNH2PARP1CHRM1GRM2HTR3A
SCHEMBL7257413 0.82 PARP1 (0.36) KCNH2PARP1GRM2HTR3ACRHR1
SCHEMBL6508880 0.81 CCR4 (0.39) HRH1CYP2D6PARP1PDCD1CD274
SCHEMBL6630822 0.80 PARP1 (0.34) HRH1KCNH2CYP2D6PARP1CHRM1
SCHEMBL7257414 0.80 KCNH2 (0.39) KCNH2PARP1GRM2HTR3A
SCHEMBL6505984 0.80 PARP1 (0.36) CYP2D6PARP1CRHR1
Hydrochloric Acid SCHEMBL6508148 0.79 PARP1 (0.36) KCNH2PARP1GRM2HTR3A
SCHEMBL6630805 0.79 PARP1 (0.43) PARP1HTR6HTR3A
SCHEMBL6631361 0.79 HDAC6 (0.46) KCNH2PARP1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309594-B1 BENZIMIDAZOLE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI AVENTIS (FR) 2004-12-15 EP claimed