SCHEMBL7258134

SCHEMBL7258134

CN(C)CCn1ccc2ccc(-c3ccccn3)cc21

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 0.67
HTR2A P28223 3/20 0.56
HTR2C P28335 3/20 0.56
BPTF Q12830 2/20 0.47
HTR6 P50406 2/20 0.46
BRD4 O60885 1/20 0.43
NOS3 P29474 2/20 0.43
NOS1 P29475 2/20 0.43
IRAK4 Q9NWZ3 1/20 0.42
NOS2 P35228 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7256762 0.73 HTR1D (0.64) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL7253051 0.73 HTR1D (0.67) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL4060777 0.73 HTR2C (1.00) HTR1DHTR2AHTR2CHTR6
SCHEMBL23479923 0.73 HTR6 (0.41) HTR2AHTR2CHTR6BRD4
Hydrochloric Acid SCHEMBL31096553 0.72 HTR6 (0.40) HTR2AHTR2CHTR6BRD4
SCHEMBL7253092 0.72 HTR1D (1.00) HTR1DHTR2AHTR2CBPTFHTR6
Hydrochloric Acid SCHEMBL23202482 0.72 HTR6 (0.40) HTR2AHTR2CHTR6BRD4
SCHEMBL7252922 0.71 HTR2A (0.64) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL23956080 0.71 HTR2C (0.69) HTR1DHTR2AHTR2CHTR6NOS3
SCHEMBL1122347 0.71 HTR2C (0.64) HTR1DHTR2AHTR2CHTR6NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine NPS ALLEXLIX CORP. 2002-11-14 US claimed
US-6635639-B2 Treatment or diagnosis of central nervous system conditions NPS ALLELIX CORP. (CA) 2003-10-21 US disclosed
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine NPS ALLEXLIX CORP. 2002-11-14 US disclosed
US-6380242-B1 FOR DIAGNOSIS AND THERAPY OF CENTRAL NERVOUS SYSTEM CONDITIONS NPS ALLELIX CORP. (CA) 2002-04-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine CNR1, CNR2, KCNH1 HTR1D 128/4885HTR2A 425/4885HTR2C 127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.