SCHEMBL7258152

SCHEMBL7258152

O=C(NCc1ccc(F)cc1C(=O)N1CCOCC1)c1nc(N2CCCCS2(O)O)c2cccnc2c1O

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CALCA P06881 9/20 0.59
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
ADORA2A P29274 3/20 0.37
ADORA1 P30542 3/20 0.37
SLC40A1 Q9NP59 1/20 0.36
CCKBR P32239 1/20 0.35
TP53 P04637 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
GRM4 Q14833 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258253 0.99 CALCA (0.58) CALCAKDM4EMAPTADORA2AADORA1
SCHEMBL7258155 0.93 CALCA (0.70) CALCAKDM4EMAPTADORA2AADORA1
SCHEMBL7262555 0.89 CALCA (0.65) CALCAKDM4EADORA2AADORA1
SCHEMBL4763683 0.89 CALCA (0.64) CALCAADORA2AADORA1TP53
SCHEMBL4765294 0.89 CALCA (0.64) CALCAKDM4EADORA2AADORA1
SCHEMBL4765622 0.88 CALCA (0.63) CALCAKDM4EADORA2AADORA1
SCHEMBL4766074 0.88 CALCA (0.63) CALCAADORA2AADORA1TP53
SCHEMBL4767331 0.88 CALCA (0.63) CALCAADORA2AADORA1TP53
Water SCHEMBL6250506 0.87 CALCA (0.62) CALCAADORA2AADORA1TP53
SCHEMBL4763116 0.87 CALCA (0.62) CALCAADORA2AADORA1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO claimed