SCHEMBL7258155

SCHEMBL7258155

O=C(NCc1ccc(F)cc1C(=O)N1CCOCC1)c1nc(N2CCCCS2(=O)=O)c2cccnc2c1O

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CALCA P06881 9/20 0.70
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
SLC40A1 Q9NP59 1/20 0.38
ADORA2A P29274 3/20 0.37
ADORA1 P30542 3/20 0.37
GRM4 Q14833 1/20 0.36
CCKBR P32239 1/20 0.35
TP53 P04637 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258152 0.93 CALCA (0.59) CALCAKDM4EMAPTSLC40A1ADORA2A
SCHEMBL7258253 0.92 CALCA (0.58) CALCAKDM4EMAPTSLC40A1ADORA2A
SCHEMBL7258249 0.92 CALCA (0.58) CALCAKDM4EMAPTSLC40A1ADORA2A
SCHEMBL7262560 0.89 CALCA (0.77) CALCAADORA2AADORA1
SCHEMBL4763498 0.89 CALCA (0.76) CALCAADORA2AADORA1TP53
SCHEMBL4765288 0.89 CALCA (0.76) CALCAADORA2AADORA1
SCHEMBL7258270 0.87 CALCA (0.74) CALCAKDM4EADORA2AADORA1
Water SCHEMBL6250514 0.87 CALCA (0.74) CALCAADORA2AADORA1TP53
SCHEMBL4763113 0.87 CALCA (0.74) CALCAADORA2AADORA1
SCHEMBL4763114 0.86 CALCA (0.73) CALCAADORA2AADORA1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO claimed