SCHEMBL7258452

SCHEMBL7258452

O=C1c2ccccc2C(=O)N1Cc1cc2c(cc1O)OCO2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.68
PKM P14618 2/20 0.68
TSHR P16473 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
GAA P10253 5/20 0.52
HSD17B10 Q99714 2/20 0.51
HPGD P15428 3/20 0.50
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CMA1 P23946 1/20 0.44
ALOX15 P16050 1/20 0.44
HTT P42858 1/20 0.44
RECQL P46063 1/20 0.43
CASP3 P42574 1/20 0.43
TGFBR1 P36897 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1080825 0.82 KMT2A (0.63) KMT2APKMTSHRSMN1; SMN2GAA
SCHEMBL19500873 0.81 KMT2A (1.00) KMT2APKMTSHRSMN1; SMN2GAA
SCHEMBL19667559 0.77 KMT2A (0.57) KMT2APKMTSHRSMN1; SMN2GAA
SCHEMBL15624560 0.74 MPO (0.50) KMT2APKMTSHRGAAHSD17B10
SCHEMBL7258443 0.73 KMT2A (0.52) KMT2APKMTSHRSMN1; SMN2HSD17B10
SCHEMBL6076008 0.73 GRM5 (0.62) KMT2ASMN1; SMN2GAAHSD17B10HPGD
SCHEMBL29195354 0.72 KMT2A (0.82) KMT2APKMTSHRSMN1; SMN2GAA
SCHEMBL6944267 0.72 KMT2A (0.83) KMT2APKMTSHRSMN1; SMN2HPGD
SCHEMBL281216 0.72 SCN9A (0.53) KMT2APKMTSHRSMN1; SMN2GAA
SCHEMBL31751934 0.71 KMT2A (0.65) KMT2AHPGDMEN1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067935-B1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) UNIV CALIFORNIA (US) 2003-08-20 EP disclosed
EP-1067935-A4 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) UNIV CALIFORNIA (US) 2001-10-04 EP disclosed
EP-1067935-A1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) The Regents of the University of California (US) 2001-01-17 EP disclosed
US-6124278-A COGNITION ACTIVATORS FOR LEARNING/MEMORY ENHANCEMENT AND TREATMENT OF BRAIN/PSYCHOLOGICAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-09-26 US disclosed
WO-1999051240-A1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1999-10-14 WO disclosed