SCHEMBL7258443

SCHEMBL7258443

CCOCOc1cc2c(cc1CN1C(=O)c3ccccc3C1=O)OCO2

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.52
PKM P14618 1/20 0.52
TSHR P16473 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
RXFP1 Q9HBX9 1/20 0.43
HPGD P15428 4/20 0.42
HSD17B10 Q99714 1/20 0.41
MAPT P10636 3/20 0.40
ALDH1A1 P00352 2/20 0.40
RPS6KA2 Q15349 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TGFBR1 P36897 1/20 0.39
RECQL P46063 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262450 0.94 KMT2A (0.45) KMT2APKMTSHRSMN1; SMN2RXFP1
SCHEMBL7263664 0.84 RXFP1 (0.39) KMT2APKMTSHRSMN1; SMN2RXFP1
SCHEMBL1080825 0.73 KMT2A (0.63) KMT2APKMTSHRSMN1; SMN2HPGD
SCHEMBL7258452 0.73 KMT2A (0.68) KMT2APKMTSHRSMN1; SMN2HPGD
SCHEMBL7262414 0.73 ALDH1A1 (0.35) KMT2ATSHRSMN1; SMN2HPGDHSD17B10
SCHEMBL19500873 0.69 KMT2A (1.00) KMT2APKMTSHRSMN1; SMN2HPGD
SCHEMBL7258246 0.66 RAB9A (0.35) KMT2ASMN1; SMN2HPGDMAPTALDH1A1
SCHEMBL3802555 0.65 PKM (0.68) KMT2APKMTSHRSMN1; SMN2RXFP1
SCHEMBL1856211 0.65 KMT2A (0.49) KMT2APKMTSHRSMN1; SMN2RXFP1
SCHEMBL1856209 0.65 KMT2A (0.49) KMT2APKMTSHRSMN1; SMN2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067935-B1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) UNIV CALIFORNIA (US) 2003-08-20 EP disclosed
EP-1067935-A4 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) UNIV CALIFORNIA (US) 2001-10-04 EP disclosed
EP-1067935-A1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) The Regents of the University of California (US) 2001-01-17 EP disclosed
US-6124278-A COGNITION ACTIVATORS FOR LEARNING/MEMORY ENHANCEMENT AND TREATMENT OF BRAIN/PSYCHOLOGICAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-09-26 US disclosed
WO-1999051240-A1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1999-10-14 WO disclosed