SCHEMBL7258658

SCHEMBL7258658

O=C(NCc1[c]cccc1)c1nc(N2CCCCS2(=O)=O)c2cccnc2c1O

nearest known ligand 0.78

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CALCA P06881 13/20 0.78
EGLN1 Q9GZT9 1/20 0.35
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
HTR6 P50406 1/20 0.33
SLC40A1 Q9NP59 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258667 0.92 CALCA (0.65) CALCAEGLN1ADORA3ADORA2AADORA2B
SCHEMBL29393055 0.84 CALCA (1.00) CALCA
SCHEMBL1198641 0.84 CALCA (1.00) CALCA
SCHEMBL7257885 0.83 CALCA (0.81) CALCAEGLN1ADORA3ADORA2AADORA2B
SCHEMBL6046599 0.83 CALCA (1.00) CALCAEGLN1
SCHEMBL968119 0.83 CALCA (0.78) CALCA
SCHEMBL4763118 0.83 CALCA (0.77) CALCAEGLN1ADORA3ADORA2AADORA2B
SCHEMBL7262566 0.82 CALCA (0.76) CALCAADORA3ADORA2AADORA2BADORA1
SCHEMBL4062690 0.81 CALCA (0.75) CALCAADORA3ADORA2AADORA2BADORA1
SCHEMBL7263607 0.81 CALCA (0.79) CALCAADORA3ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO disclosed