SCHEMBL7258667

SCHEMBL7258667

O=C(NCc1[c]cccc1)c1nc(N2CCCCS2(O)O)c2cccnc2c1O

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CALCA P06881 9/20 0.65
EGLN1 Q9GZT9 2/20 0.35
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2B P29275 1/20 0.33
HTR6 P50406 1/20 0.33
TP53 P04637 1/20 0.33
ALOX15 P16050 1/20 0.33
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32
MCL1 Q07820 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258658 0.92 CALCA (0.78) CALCAEGLN1ADORA2AADORA1ADORA3
SCHEMBL4063925 0.84 CALCA (0.84) CALCATP53
SCHEMBL7257882 0.83 CALCA (0.68) CALCAEGLN1ADORA2AADORA1ADORA3
SCHEMBL6046600 0.83 CALCA (0.84) CALCAEGLN1
SCHEMBL968122 0.83 CALCA (0.64) CALCAEGLN1HTR6TP53ALOX15
SCHEMBL4763117 0.83 CALCA (0.64) CALCAEGLN1ADORA2AADORA1ADORA3
SCHEMBL7262570 0.82 CALCA (0.63) CALCAADORA2AADORA1ADORA3ADORA2B
SCHEMBL7263617 0.81 CALCA (0.67) CALCAADORA2AADORA1ADORA3ADORA2B
SCHEMBL7262169 0.81 CALCA (0.62) CALCAEGLN1ADORA2AADORA1ADORA3
SCHEMBL4062694 0.81 CALCA (0.62) CALCAADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO disclosed