SCHEMBL7258794

SCHEMBL7258794

CN(C)C(=O)c1cc(F)ccc1CNC(=O)c1ncc2cccnc2c1O

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.45
ADORA1 P30542 6/20 0.45
EGLN1 Q9GZT9 7/20 0.43
CALCA P06881 3/20 0.38
PIK3CD O00329 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262269 0.89 ADORA2A (0.47) ADORA2AADORA1EGLN1CALCA
SCHEMBL7258671 0.86 ADORA2A (0.44) ADORA2AADORA1EGLN1CALCA
SCHEMBL4766011 0.81 ADORA2A (0.42) ADORA2AADORA1EGLN1CALCA
SCHEMBL7262168 0.81 ADORA2A (0.43) ADORA2AADORA1EGLN1CALCA
SCHEMBL7258997 0.80 ADORA2A (0.42) ADORA2AADORA1EGLN1CALCA
SCHEMBL7262470 0.80 ADORA2A (0.42) ADORA2AADORA1EGLN1CALCA
SCHEMBL7258981 0.79 ADORA2A (0.41) ADORA2AADORA1EGLN1CALCA
SCHEMBL7258140 0.79 ADORA2A (0.43) ADORA2AADORA1
SCHEMBL4068615 0.78 EGLN1 (0.55) EGLN1CALCA
SCHEMBL7262304 0.76 CALCA (0.56) ADORA2AADORA1CALCAPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO claimed
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO disclosed