SCHEMBL7259046

SCHEMBL7259046

Cc1cccc(CBr)c1.Cc1cccc(CN2CCC(CNC(=O)c3cc(Cl)c(N)[nH]c3=O)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.49
CXCR4 P61073 5/20 0.49
HTR4 Q13639 3/20 0.48
DRD2 P14416 3/20 0.47
DRD4 P21917 3/20 0.47
DRD3 P35462 2/20 0.47
CCR2 P41597 1/20 0.47
KCNH2 Q12809 1/20 0.47
CACNA1I Q9P0X4 1/20 0.47
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
THRB P10828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6328378 0.96 CXCR4 (0.52) HTTCXCR4HTR4DRD2DRD4
SCHEMBL7259058 0.90 KCNH2 (0.56) HTTHTR4DRD2DRD4DRD3
SCHEMBL7254037 0.90 HTR4 (0.51) HTTHTR4DRD2DRD4DRD3
SCHEMBL6328740 0.87 HDAC3 (0.50) HTTHTR4DRD2DRD4DRD3
SCHEMBL6329054 0.87 TP53 (0.57) HTTCXCR4HTR4DRD2DRD4
SCHEMBL6329791 0.87 KCNH2 (0.61) HTTHTR4DRD2DRD4DRD3
SCHEMBL6329006 0.87 HTR4 (0.52) HTTHTR4DRD2DRD4DRD3
SCHEMBL6329269 0.87 DRD2 (0.58) HTR4DRD2DRD4DRD3
SCHEMBL6336358 0.85 HTR4 (0.56) HTR4DRD2DRD4DRD3
SCHEMBL7257582 0.85 HTR4 (0.61) HTR4DRD2DRD4DRD3CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003057688-A2 OXO OR OXY-PYRIDINE COMPOUNDS AS 5-HT4 RECEPTOR MODULATORS PFIZER JAPAN INC. (JP) 2003-07-17 WO disclosed