SCHEMBL7259092

SCHEMBL7259092

CC(=O)c1cc(-c2ccccc2)nnc1Cl

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 16/20 0.71
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
RAB9A P51151 1/20 0.47
HSD17B10 Q99714 1/20 0.47
PPARA Q07869 1/20 0.43
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
PDE10A Q9Y233 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL580314 0.86 CASP1 (0.76) CASP1SMN1; SMN2ALDH1A1HSD17B10PPARA
SCHEMBL7255594 0.84 CASP1 (0.53) CASP1SMN1; SMN2NPC1ALDH1A1HPGD
SCHEMBL1752817 0.83 CASP1 (1.00) CASP1KDM4E
SCHEMBL7255661 0.82 CASP1 (0.69) CASP1ALDH1A1
SCHEMBL27225888 0.75 CASP1 (0.56) CASP1SMN1; SMN2ALDH1A1HSD17B10KDM4E
SCHEMBL30850823 0.75 CASP1 (0.56) CASP1SMN1; SMN2ALDH1A1HSD17B10KDM4E
SCHEMBL7255590 0.73 CASP1 (0.57) CASP1
SCHEMBL581917 0.73 CASP1 (0.53) CASP1SMN1; SMN2NPC1ALDH1A1HPGD
SCHEMBL30962961 0.73 CASP1 (0.53) CASP1SMN1; SMN2NPC1ALDH1A1HPGD
SCHEMBL530338 0.73 CASP1 (0.57) CASP1SMN1; SMN2NPC1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003080616-A1 PYRAZOLOPYRIDAZINE DERIVATIVES, PROCESS FOR PREPARATION AND USE FOR THE INHIBITION OF GSK-3 GLAXO GROUP LIMITED (GB) 2003-10-02 WO disclosed