SCHEMBL7259291

SCHEMBL7259291

O=C(Nc1ccc2[nH]ncc2c1)c1cc(NCCc2ccccn2)c(F)cc1F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 7/20 0.58
GRK2 P25098 2/20 0.58
GRK5 P34947 2/20 0.58
JAK2 O60674 3/20 0.55
JAK1 P23458 2/20 0.55
GRK1 Q15835 1/20 0.51
NPC1 O15118 6/20 0.51
RAB9A P51151 6/20 0.51
HPGD P15428 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MAOB P27338 2/20 0.48
ROCK2 O75116 5/20 0.48
DYRK3 O43781 1/20 0.48
MAP4K4 O95819 1/20 0.48
RPS6KB1 P23443 1/20 0.48
CLK2 P49760 1/20 0.48
CSNK2A1 P68400 1/20 0.48
DYRK1A Q13627 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7255625 0.94 NPC1 (0.57) ROCK1GRK2GRK5JAK2JAK1
SCHEMBL7256998 0.91 JAK2 (0.56) ROCK1GRK2GRK5JAK2JAK1
SCHEMBL7255709 0.84 JAK2 (0.58) ROCK1JAK2JAK1NPC1RAB9A
SCHEMBL7255808 0.81 JAK2 (0.57) ROCK1JAK2JAK1NPC1RAB9A
SCHEMBL7255640 0.78 JAK2 (0.52) ROCK1GRK2GRK5JAK2JAK1
SCHEMBL7259294 0.78 NPC1 (0.50) ROCK1GRK2GRK5JAK2JAK1
SCHEMBL7261177 0.77 JAK2 (0.48) ROCK1GRK2GRK5JAK2JAK1
SCHEMBL7256698 0.77 NPC1 (0.61) ROCK1JAK2JAK1NPC1RAB9A
SCHEMBL7261149 0.77 NPC1 (0.68) ROCK1JAK2JAK1NPC1RAB9A
SCHEMBL7256479 0.76 LRRK2 (0.53) ROCK1JAK2JAK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003002518-A1 NOVEL 2,4-DIFLUOROBENZAMIDE DERIVATIVES AS ANTIVIRAL AGENTS DONG HWA PHARM. IND. CO., LTD. (KR) 2003-01-09 WO disclosed