SCHEMBL7259294

SCHEMBL7259294

Nc1c(F)c(CCc2ccccn2)cc(C(=O)Nc2ccc3[nH]ncc3c2)c1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
JAK2 O60674 5/20 0.50
ROCK1 Q13464 5/20 0.50
JAK1 P23458 4/20 0.50
GRK2 P25098 2/20 0.50
GRK5 P34947 2/20 0.50
GRK1 Q15835 1/20 0.47
ROCK2 O75116 2/20 0.47
DYRK3 O43781 1/20 0.47
MAP4K4 O95819 1/20 0.47
RPS6KB1 P23443 1/20 0.47
CLK2 P49760 1/20 0.47
CSNK2A1 P68400 1/20 0.47
DYRK1A Q13627 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
MAOB P27338 2/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7255631 0.93 RAB9A (0.55) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL7257003 0.92 NPC1 (0.51) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL7255642 0.80 TRPV1 (0.49) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL7259291 0.78 ROCK1 (0.58) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL7256998 0.76 JAK2 (0.56) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL7256506 0.75 LRRK2 (0.49) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL15764656 0.72 NPC1 (0.81) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL7255625 0.72 NPC1 (0.57) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL16888856 0.71 NPC1 (0.64) NPC1RAB9AJAK2ROCK1JAK1
SCHEMBL7261242 0.71 NPC1 (0.48) NPC1RAB9AMAP4K4CLK2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003002518-A1 NOVEL 2,4-DIFLUOROBENZAMIDE DERIVATIVES AS ANTIVIRAL AGENTS DONG HWA PHARM. IND. CO., LTD. (KR) 2003-01-09 WO disclosed