SCHEMBL7259883

SCHEMBL7259883

CN(CCCCI)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 2/20 0.40
HDAC6 Q9UBN7 2/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
CTSK P43235 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.33
PDK2 Q15119 1/20 0.33
LMNA P02545 1/20 0.33
GBA1 P04062 1/20 0.32
METAP2 P50579 1/20 0.32
TRPV4 Q9HBA0 1/20 0.31
FPR3 P25089 1/20 0.31
FPR2 P25090 1/20 0.31
CACNA1G O43497 1/20 0.30
CACNA1B Q00975 1/20 0.30
CACNA1C Q13936 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA7 P43166 1/20 0.30
AAK1 Q2M2I8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22940133 0.98 HDAC6 (0.39) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL5563929 0.94 HDAC6 (0.38) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL4613481 0.86 HDAC6 (0.36) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL25720861 0.83 ALDH1A1 (0.42) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL2478206 0.83 TDP1 (0.44) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL3161597 0.83 CA14 (0.41) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL8476324 0.83 CA14 (0.41) CA14HDAC6HDAC1HDAC2L3MBTL1
SCHEMBL10260946 0.82 HDAC6 (0.40) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL25236870 0.81 CA14 (0.43) CA14HDAC6HDAC1HDAC2CTSK
SCHEMBL12281742 0.81 TDP1 (0.47) CA14HDAC6HDAC1HDAC2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine INSILICO MEDICINE IP LIMITED (HK) 2025-05-08 US disclosed
WO-2024260325-A1 SYNTHESIS OF MACROCYCLIC COMPOUND AND MEDICAL USE OF MACROCYCLIC COMPOUND 英矽智能科技知识产权有限公司 2024-12-26 WO disclosed
EP-4455132-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE Insilico Medicine IP Limited (HK) 2024-10-30 EP disclosed
WO-2023116761-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 英矽智能科技知识产权有限公司 2023-06-29 WO disclosed
WO-2023116761-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 英矽智能科技知识产权有限公司 2023-06-29 WO disclosed
EP-3327016-B1 PREPARATION OF MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2021-06-16 EP disclosed
EP-3327016-A1 PREPARATION OF MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2018-05-30 EP disclosed
EP-3091011-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2017-12-27 EP disclosed
US-9758510-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-09-12 US disclosed
WO-2003013526-A1 ANTICOAGULANT COMPOUNDS MERCK & CO. INC. (US) 2003-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine DPYD, TYMP, NUDT1 CA14 2694/4885HDAC6 1013/4885HDAC1 1255/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.