SCHEMBL7260498

SCHEMBL7260498

O=C(O)c1ccc(CNc2nc(OCc3ccccc3)nc3ccc(Cl)cc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.54
CNR2 P34972 5/20 0.50
PDE5A O76074 4/20 0.50
HTR3A P46098 1/20 0.49
HRH4 Q9H3N8 1/20 0.49
PPARA Q07869 1/20 0.47
RXRA P19793 1/20 0.46
RXRB P28702 1/20 0.46
RXRG P48443 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254764 0.81 CNR1 (0.57) CNR1PDE5AHTR3AHRH4
SCHEMBL7260274 0.80 CNR1 (0.56) CNR1PDE5AHTR3AHRH4
SCHEMBL15905004 0.76 PPARA (0.50) PPARA
SCHEMBL7258507 0.74 HRH4 (0.55) CNR1HTR3AHRH4
SCHEMBL2590769 0.73 RAD52 (0.68) PDE5AHTR3AHRH4
SCHEMBL3638867 0.73 PDE5A (0.73) PDE5AHTR3AHRH4
SCHEMBL7254637 0.73 CNR1 (0.58) CNR1CNR2PDE5AHTR3AHRH4
SCHEMBL8670004 0.73 EGFR (0.57) CNR1PDE5A
SCHEMBL15905225 0.72 PPARA (0.63) PPARAMRGPRX4
SCHEMBL7497383 0.72 PDE5A (0.59) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055866-A1 QUINAZOLINE AND QUINOLINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO disclosed