SCHEMBL7260274

SCHEMBL7260274

O=C(O)c1ccc(CNc2nc(O)nc3ccc(Cl)cc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.56
CTNNB1 P35222 7/20 0.49
TCF7L2 Q9NQB0 7/20 0.49
PDE5A O76074 4/20 0.49
ALDH1A1 P00352 1/20 0.49
HRH4 Q9H3N8 4/20 0.46
HTR3A P46098 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254764 0.89 CNR1 (0.57) CNR1CTNNB1TCF7L2PDE5AALDH1A1
SCHEMBL7260498 0.80 CNR1 (0.54) CNR1PDE5AHRH4HTR3A
SCHEMBL7258507 0.79 HRH4 (0.55) CNR1CTNNB1TCF7L2ALDH1A1HRH4
SCHEMBL7254637 0.78 CNR1 (0.58) CNR1CTNNB1TCF7L2PDE5AALDH1A1
SCHEMBL7503857 0.77 PDE5A (0.69) PDE5AALDH1A1
SCHEMBL7260501 0.74 CTNNB1 (0.65) CNR1CTNNB1TCF7L2
SCHEMBL27840330 0.74 PDE5A (0.53) CNR1PDE5AALDH1A1
SCHEMBL7258119 0.73 FABP3 (0.53) CNR1CTNNB1TCF7L2ALDH1A1
SCHEMBL2590769 0.72 RAD52 (0.68) PDE5AALDH1A1HRH4HTR3A
SCHEMBL3638867 0.72 PDE5A (0.73) PDE5AALDH1A1HRH4HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055866-A1 QUINAZOLINE AND QUINOLINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO disclosed