SCHEMBL7260682

SCHEMBL7260682

N=C(N)Nc1cccc(CC(N)C(=O)O)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.70
NOS1 P29475 3/20 0.70
NOS2 P35228 3/20 0.70
SLC7A5 Q01650 8/20 0.54
PTGS1 P23219 2/20 0.54
ALPI P09923 1/20 0.54
PKM P14618 1/20 0.54
XIAP P98170 1/20 0.54
GRIA2 P42262 1/20 0.52
CASR P41180 1/20 0.48
KDM4E B2RXH2 1/20 0.48
USP2 O75604 1/20 0.48
EGFR P00533 1/20 0.48
LCK P06239 1/20 0.48
FYN P06241 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
ALOX15 P16050 1/20 0.48
HTR2A P28223 1/20 0.48
PTGS2 P35354 1/20 0.48
RECQL P46063 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL288850 1.00 NOS3 (0.70) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL29589136 1.00 NOS3 (0.70) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL287831 1.00 NOS3 (0.70) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL20715034 0.89 NOS3 (0.59) NOS3NOS1NOS2SLC7A5GRIA2
SCHEMBL6046229 0.87 NOS3 (0.71) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL4629196 0.86 NOS3 (0.53) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL3152192 0.85 NOS3 (0.73) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL20502934 0.85 NOS3 (0.73) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL20502933 0.85 NOS3 (0.73) NOS3NOS1NOS2SLC7A5PTGS1
SCHEMBL8075751 0.83 NOS3 (0.50) NOS3NOS1NOS2CASRITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874472-A Aminoacid derivatives as no synthase inhibitors GLAXO WELLCOME INC. (US) 1999-02-23 US claimed
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP claimed
EP-0705257-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-04-10 EP claimed
WO-1995000505-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-01-05 WO claimed
EP-4724459-A1 PEPTIDE COMPOSITIONS TARGETING GLYPICAN-3 AND USES THEREOF Peptidream Inc (JP) 2026-04-15 EP disclosed
EP-4724457-A2 RADIOPHARMACEUTICAL COMPOSITIONS TARGETING GLYPICAN-3 AND USES THEREOF Rayzebio, Inc. (US) 2026-04-15 EP disclosed
WO-2024254339-A9 RADIOPHARMACEUTICAL COMPOSITIONS TARGETING GLYPICAN-3 AND USES THEREOF RAYZEBIO, INC. (US) 2025-10-16 WO disclosed
WO-2024252336-A1 PEPTIDE COMPOSITIONS TARGETING GLYPICAN-3 AND USES THEREOF PEPTIDREAM INC. (JP) 2024-12-12 WO disclosed
WO-2024254339-A2 RADIOPHARMACEUTICAL COMPOSITIONS TARGETING GLYPICAN-3 AND USES THEREOF RAYZEBIO, INC. (US) 2024-12-12 WO disclosed
US-20240010627-A1 NOVEL GUANIDINE DERIVATIVE AND METHOD FOR PRODUCING SAME PEPTIDREAM INC. (JP) 2024-01-11 US disclosed
US-20230391828-A1 REGULATORS OF CELL DIVISION TECHNISCHE UNIVERSITAT DRESDEN (DE) 2023-12-07 US disclosed
EP-4276096-A1 NOVEL GUANIDINE DERIVATIVE AND METHOD FOR PRODUCING SAME PeptiDream Inc. (JP) 2023-11-15 EP disclosed
WO-2022149610-A1 NOVEL GUANIDINE DERIVATIVE AND METHOD FOR PRODUCING SAME ペプチドリーム株式会社 2022-07-14 WO disclosed
EP-3981784-A1 REGULATORS OF CELL DIVISION Technische Universität Dresden (DE) 2022-04-13 EP disclosed
US-6649593-B1 Amino acid derivatives including serine, leucine, valine, arginine, asparginine, methionine, glycine and phenylalanine units; S1 protease inhibition; modulation of cholesterol homeostasis in cells TULARIK INC. 2003-11-18 US disclosed
WO-2001027138-A2 MODULATORS OF SREBP PROCESSING TULARIK INC. (US) 2001-04-19 WO disclosed
US-5874472-A Aminoacid derivatives as no synthase inhibitors GLAXO WELLCOME INC. (US) 1999-02-23 US disclosed
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed
EP-0705257-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-04-10 EP disclosed
WO-1995000505-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230391828-A1 REGULATORS OF CELL DIVISION PCNA, BOD1L1, MKI67 NOS3 3629/4885NOS1 3182/4885NOS2 3515/4885
US-20240010627-A1 NOVEL GUANIDINE DERIVATIVE AND METHOD FOR PRODUCING SAME GMPS, MAPT, UROD NOS3 599/4885NOS1 351/4885NOS2 305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.